SR 144528

Tocris Bioscience

Product Information

Product Overview:

High affinity and selective CB 2 inverse agonist (K i = 0.6 nM). Exhibits >700-fold selectivity for CB 2 over CB 1 receptors. Blocks the effects of CP 55,940 (Cat. No. 0949) on forskolin-sensitive adenylyl cyclase activity and MAPK in CHO cells expressing CB 2 receptors. Also blocks CP 55,940-induced B-cell activation. Orally bioavailable.

Catalog#: 5039-10MG
LID#: 4129904B
Quantity :
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Chemical Name5-(4-Chloro-3-methylphenyl)-1-[(4-m?ethylphenyl)methyl]-N-[(1S,2S,4R)-1,3,3-trimethylb?icyclo[2.2.1]hept-2-yl]-1H-pyrazole-3-carboxamide
SolubilitySoluble to 100 mM in DMSO and to 100 mM in ethanol
Molecular Weight476.05
Grade/Purity>98 %
Chemical FormulaC29H34ClN3O
Unit Size10mg
Safety StatementsThe technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Sample AvailabilityNo

Shipping & Handling

Estimated Ship Time: 3 Business Days

Shipped In: Dry Ice

Hazardous Material: No


Storage Temperature: Store at -20°C

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